D. Phil and Post-doctoral Publications (with Prof. Steve Davies)

96. Strategies for the construction of morphinan alkaloid AB-rings: regioselective Friedel-Crafts-type cyclisations of γ-aryl-β-benzoylamido acids with asymmetrically substituted γ-aryl rings

S. G. Davies, E. C. Goddard, P. M Roberts, A. J. Russell, A. D. Smith, J. E. Thomson, J. M. Withey

Tetrahedron: Asymmetry201627, 274-284

95. Asymmetric synthesis of piperidines and octahydroindolizines using a one-pot ring-closure/N-debenzylation procedure

S. G. Davies, A. M. Fletcher, D. G. Hughes, J. A. Lee, P. D. Price, P. M. Roberts, A. J. Russell, A. D. Smith, J. E. Thomson and O. M. H. Williams

Tetrahedron201167, 9975-9992

94. Asymmetric Synthesis of syn- and anti-α-deuterio-β3-phenylalanine derivatives

S. G. Davies, E. M. Foster, C. R. McIntosh, P. M. Roberts, T. E. Rosser, A. D. Smith and J. E. Thomson

Tetrahedron: Asymmetry201122, 1035-1050

93. A systematic study of the solid state and solution phase conformational preferences of β-peptides derived from C(3)-alkyl substituted transpentacin derivatives

E. Abraham, T. D. W. Claridge, S. G. Davies, B. Odell, P. M. Roberts, A. J. Russell, A. D. Smith, L. J. Smith, H. R. Storr, M. J. Sweet, A. L Thompson, J. E. Thomson, G. E. Tranter and D. J. Watkin

Tetrahedron: Asymmetry201122, 69-100

92. A systematic study of the solid state and solution phase conformational preferences of β-peptides derived from transpentacin

E. Abraham, C. W. Bailey, T. D. W. Claridge, S. G. Davies, K. B. Ling, B. Odell, T. L. Rees, P. M. Roberts, A. J. Russell, A. D. Smith, L. J. Smith, H. R. Storr, M. J. Sweet, A. L. Thompson, J. E. Thomson, G. E. Tranter and D. J. Watkin

Tetrahedron: Asymmetry201021, 1797-1815

91. Doubly diastereoselective conjugate addition of enantiopure lithium amides to enantiopure N-enoyl oxazolidin-2-ones: a mechanistic probe

S. G. Davies, A. M. Fletcher, G. J. Hermann, G. Poce, P. M. Roberts, A. D. Smith, M. J. Sweet and J. E. Thomson

Tetrahedron: Asymmetry201021, 1635-1648

90. Alkylation and aldol reactions of acyl derivatives of N-1-(1′-naphthyl)ethyl-O-tert-butylhydroxylamine: asymmetric synthesis of α-alkoxy-, α-substituted-β-alkoxy- and α,β-dialkoxyaldehydes

A. N. Chernega, S. G. Davies, A. M. Fletcher, C. J. Goodwin, D. Hepworth, R. S. Prasad, P. M. Roberts, E. D. Savory, A. D. Smith and J. E. Thomson

Tetrahedron201066, 4167-4194

89. Asymmetric Synthesis of Piperidines and Octahydroindolizines

S. G. Davies, D. G. Hughes, P. D. Price, P. M. Roberts, A. J. Russell, A. D. Smith, J. E. Thomson and O. M. H. Williams

Synlett2010, 567-570

88. Asymmetric synthesis of Sedum alkaloids via lithium amide conjugate addition

S. G. Davies, A. M. Fletcher, P. M. Roberts and A. D. Smith

Tetrahedron200965, 10192-10213

87. The dienolate aldol reaction of (E)-N-crotonoyl C(4)-isopropyl SuperQuat: asymmetric synthesis of α-vinyl-β-hydroxycarboxylic acid derivatives and conversion to α-ethylidene-β-hydroxyesters (β-substituted Baylis-Hillman products)

S. G. Davies, D. L. Elend, S. Jones, P. M. Roberts, E. D. Savory, A. D. Smith and J. E. Thomson

Tetrahedron200965, 7837-7851

86. Ammonium-directed oxidation of cyclic allylic and homoallylic amines

C. W. Bond, A. J. Cresswell, S. G. Davies, W. Kurosawa, J. A. Lee, A. M. Fletcher, P. M. Roberts, A. J. Russell, A. D. Smith and J. E. Thomson

J. Org. Chem200974, 6735-6748

85. Doubly diastereoselective [3,3]-sigmatropic aza-Claisen rearrangements

S. G. Davies, A. C. Garner, R. L. Nicholson, J. Osborne, P. M. Roberts, E. D. Savory, A. D. Smith and J. E. Thomson

Org. Biomol. Chem.20097, 2604-2611

84. Iodine-mediated ring-closing iodoamination with concomitant N-debenzylation for the asymmetric synthesis of polyhydroxylated pyrrolidines

S. G. Davies, R. L. Nicholson, P. D. Price, P. M. Roberts, A. J. Russell, E. D. Savory, A. D. Smith, and J. E. Thomson

Tetrahedron: Asymmetry200920, 758-772

83. A Tandem Conjugate Addition/Cyclization Protocol for the Asymmetric Synthesis of 2-Aryl-4-aminotetrahydroquinoline-3-carboxylic Acid Derivatives

S. G. Davies, N. Mujtaba, P. M. Roberts, A. D. Smith and J. E. Thomson

Org. Lett.200911, 1959-1962

82. Double diastereoselective conjugate addition of homochiral lithium amides to homochiral cis- and trans-γ,δ-dioxolane-containing α,β-unsaturated esters

S. G. Davies, M. J. Durbin, E. C. Goddard, P. M. Kelly, W. Kurosawa, J. A. Lee, R. L. Nicholson, P. D. Price, P. M. Roberts, A. J. Russell, P. M. Scott and A. D. Smith

Org. Biomol. Chem.20097, 761-776

81. Stereoselective functionalisation of cis- and trans-2-ferrocenyl-3-pivaloyl-1,3-oxazolidin-5-ones; asymmetric synthesis of (R)- and (S)-2-alkyl-2-aminopent-4-enoic acids and (2R,3S)-2-amino-3-hydroxy-2-methyl-3-phenylpropanoic acid

F. Alonso, S. G. Davies, A. S. Elend, M. A. Leech, P. M. Roberts, A. D. Smith and J. E. Thomson

Org. Biomol. Chem.20097, 527-536

80. Kinetic and thermodynamic control in the stereoselective formation of trans- and cis-4-alkyl-2-ferrocenyl-3-pivaloyl-1,3-oxazolidin-5-ones

F. Alonso, S. G. Davies, A. S. Elend and A. D. Smith

Org. Biomol. Chem.20097, 518-526

79. Parallel kinetic resolution of tert-butyl (RS)-6-alkyl-cyclohex-1-ene-carboxylates for the asymmetric synthesis of 6-alkyl-substituted cishexacin derivatives

S. G. Davies, M. J. Durbin, S. J. S. Hartman, A. Matsuno, P. M. Roberts, A. J. Russell, P. M. Scott, A. D. Smith, J. E. Thomson and S. M. Toms

Tetrahedron: Asymmetry200819, 2870-2881

78. Highly (E)-selective Wadsworth-Emmons reactions promoted by methylmagnesium bromide

T. D. W. Claridge, S. G. Davies, J. A. Lee, R. L. Nicholson, P. M. Roberts, A. J. Russell, A. D. Smith and S. M. Toms

Org. Lett.200810, 5437-5440

77. Pure by NMR?

T. D. W. Claridge, S. G. Davies, M. E. C. Polywka, P. M. Roberts, A. J. Russell, E. D. Savory and A. D. Smith

Org. Lett.200810, 5433-5436

76. Ammonium-directed dihydroxylation: metal-free synthesis of the diastereoisomers of 3-aminocyclohexane-1,2-diol

C. Aciro, S. G. Davies, P. M. Roberts, A. J. Russell, A. D. Smith and J. E. Thomson

Org. Biomol. Chem.20086, 3762

75. Stereoselective functionalisation of SuperQuat enamides: asymmetric synthesis of homochiral 1,2-diols and α-benzyloxy carbonyl compounds

C. Aciro, S. G. Davies, A. C. Garner, Y. Ishii, M-S. Key, K. B. Ling, R. S. Prasad, P. M. Roberts, H. Rodriguez-Solla, C. O’Leary-Steele, A. J. Russell, H. J. Sanganee, E. D. Savory, A. D. Smith, J. E. Thomson

Tetrahedron, 200864, 9320

74. Parallel kinetic resolution oftert-butyl (RS)-3-oxy-substituted cyclopent-1-ene-carboxylates for the asymmetric synthesis of 3-oxy-substituted cispentacin and transpentacin derivatives

Y. Aye, S. G. Davies, A. C. Garner, P. M. Roberts, A. D. Smith and J. E. Thomson

Org. Biomol. Chem.20086, 2195

73. Asymmetric synthesis ofN,O,O,O-tetra-acetyl D-lyxo-phytosphingosine, jaspine B (pachastrissamine) and its C(2)-epimer, and deoxoprosophyllinevialithium amide conjugate addition

E. Abraham, E. A. Brock, J. I. Candela-Lena, S. G. Davies, M. Georgiou, R. L. Nicholson, J. H. Perkins, P. M. Roberts, A. J. Russell, E. M. Sánchez-Fernández, P. M. Scott, A. D. Smith and J. E. Thomson

Org. Biomol. Chem.20086, 1665

72. Asymmetric synthesis of vicinal amino alcohols: xestoaminol C, sphinganine and sphingosine

E. Abraham, S. G. Davies, N. L. Millican, R. L. Nicholson, P. M. Roberts and A. D. Smith

Org. Biomol. Chem.20086, 1655

71. An Oxidatively Activated Safety Catch Linker for Solid Phase Synthesis

S. G. Davies, D. A. B. Mortimer, A. W. Mulvaney, A. J. Russell, H. Skarphedinsson, A. D. Smith and R. J. Vickers

Org. Biomol. Chem.20086, 1625

70. Asymmetric synthesis of N,O,O,O-tetra-acetyl D-lyxo-phytosphingosine, jaspine B (pachastrissamine) and its C(2)-epimer

E. Abraham, J. I. Candela-Lena, S. G. Davies, M. Georgiou, R. L. Nicholson, P. M. Roberts, A. J. Russell, E. M. Sanchez-Fernandez, A. D. Smith and J. E. Thomson

Tetrahedron: Asymmetry200718, 2510

69. Asymmetric synthesis of β-amino-γ-substituted-γ-butyrolactones: double diastereoselective conjugate addition of homochiral lithium amides to homochiral α,β-unsaturated esters

T. Cailleau, J. W. B. Cooke, S. G. Davies, K. B. Ling, A. Naylor, R. L. Nicholson, P. D. Price, P. M. Roberts, A. J. Russell, A. D. Smith and J. E. Thomson

Org. Biomol. Chem.2007, 5, 3922

68. Evaluating β-amino acids as enantioselective organocatalysts of the Hajos-Parrish-Eder-Sauer-Wiechert Reaction

S. G. Davies, A. J. Russell, R. L. Sheppard, A. D. Smith and J. E. Thomson

Org. Biomol. Chem.20075, 3190

67. Asymmetric Synthesis of β2-amino acids: 2-substituted-3-aminopropanoic acids fromN-acryloyl SuperQuat derivatives

J. E. Beddow, S. G. Davies, K. B. Ling, P. M. Roberts, A. J. Russell, A. D. Smith and J. E. Thomson

Org. Biomol. Chem.20075, 2812

66. Parallel Synthesis of homochiral β-amino acids

S. G. Davies, A. W. Mulvaney, A. J. Russell and A. D. Smith

Tetrahedron: Asymmetry200718, 1554

65. Asymmetric synthesis of β-substituted Baylis-Hillman products via lithium amide conjugate addition

A. Chernega, S. G. Davies, D. L. Elend, C. A. P. Smethurst, P. M. Roberts, A. D. Smith and G. D. Smyth

Tetrahedron200763, 7036

64. Conjugate addition of homochiral lithium amides to achiral γ-benzyloxy- and γ-tert-butyldimethylsilyloxy-but-2-enoates and but-2-enamides: asymmetric synthesis of 3-amino-butyrolactones

J. W. B. Cooke, S. G. Davies, A. Naylor, R. L. Nicholson, P. D. Price and A. D. Smith

Tetrahedron200763, 5855

63. Diastereoselective synthesis of quaternary α-amino acids from d iketopiperazine templates

S. G. Davies, A. C. Garner, J. V. A. Ouzman, P. M. Roberts, A. D. Smith, E. J. Snow, J. E. Thomson, J. A. Tamayo and R. J. Vickers

Org. Biomol. Chem.20075, 2138

62. Asymmetric synthesis of 3,4-anti- and 3,4-syn-substituted aminopyrrolidines via lithium amide conjugate addition

S. G. Davies, A. C. Garner, E. C. Goddard, D. Kruchinin, P. M. Roberts, A. D. Smith, H. Rodriguez-Solla, J. E. Thomson and S. M. Toms

Org. Biomol. Chem.20075, 1961

61. Asymmetric Three and [2+1] Component Conjugate Addition Reactions for the Stereoselective Synthesis of Polysubstituted Piperidinones

S. G. Davies, P. M. Roberts and A. D. Smith

Org. Biomol. Chem.20075, 1405

60. On the origins of diastereoselectivity in the alkylation of diketopiperazine enolates

S. D. Bull, S. G. Davies, A. C. Garner, A. L. Parkes, P. M. Roberts, T. G. R. Sellers, A. D. Smith, J. A. Tamayo, J. E. Thomson and R. J. Vickers

New Journal of Chemistry200731, 486

59. Homochiral Lithium Amides for the Asymmetric Synthesis of β-Amino Acids

S. G. Davies, N. M. Garrido, D. Kruchinin, O. Ichihara, L. J. Kotchie, P. D. Price, A. J. Price-Mortimer, A. J. Russell and A. D. Smith

Tetrahedron: Asymmetry200617, 1793

58. SuperQuat 5,5-Dimethyl-4-iso-propyloxazolidin-2-one as a Mimic of Evans 4-tert-butyloxazolidin-2-one

S . D. Bull, S. G. Davies, A. C. Garner, D. Kruchinin, M-S. Key, P. M. Roberts, E. D. Savory, A. D. Smith and J. E. Thomson

Org. Biomol. Chem.20064, 2945

57. Enantiodiscrimination of racemic electrophiles by diketopiperazine enolates: asymmetric synthesis of 3-methyl aspartates and methyl 2-amino-3-aryl-butanoates

S. D. Bull, S. G. Davies, S. W. Epstein, A. C. Garner, N. Mujtaba, E. D. Savory, A. D. Smith, J. A. Tamayo and D. J. Watkin

Tetrahedron200662, 7911

56. Oxazinanones as Chiral Auxiliaries: Synthesis and Evaluation in Enolate Alkylations and Aldol Reactions

S. G. Davies, A. C. Garner, P. M. Roberts, A. D. Smith, M. J. Sweet and J. E. Thomson

Org. Biomol. Chem.20064, 2753

55. Lithium Amide Conjugate Addition for the Asymmetric Synthesis of 3-Aminopyrrolidines

S. G. Davies, A. C. Garner, E. C. Goddard, D. Kruchinin, P. M. Roberts, A. D. Smith and H. Rodriguez-Solla

Chem. Commun., 2006, 2664

54. Asymmetric Synthesis of α-Mercapto-β-Amino Acid Derivatives: Application to the Synthesis of Polysubstituted Thiomorpholines

J. I. Candela-Lena, S. G. Davies, P. M. Roberts, B. Roux, A. J. Russell, E. M. Sánchez-Fernández and A. D. Smith

Tetrahedron: Asymmetry2006 , 17, 1135

53. The conjugate addition of enantiomerically pure lithium amides as homochiral ammonia equivalents: scope, limitations and synthetic applications

S. G. Davies, P. D. Price and A. D. Smith

Tetrahedron: Asymmetry200516, 2833

52. Ammonium directed dihydroxylation ofN,N-dibenzylamino-cyclohex-2-ene: metal-free syntheses of the diastereoisomers of 3-dibenzylamino-1,2-dihydroxycyclohexane

S. G. Davies, M. J. C. Long and A. D. Smith

Chem. Commun.2005, 4536

51. Highly enantioselective organocatalysis of the Hajos-Parrish-Eder-Sauer-Wiechert Reaction by the β-amino acid cispentacin

S. G. Davies, R. L. Sheppard, A. D. Smith and J. E. Thomson

Chem. Commun.2005, 3802

50. Kinetic Resolution and Parallel Kinetic Resolution of methyl (RS)-5-alkyl-cyclopentene-1-carboxylates for the asymmetric synthesis of 5-alkyl-cispentacin derivatives

S. G. Davies, A. C. Garner, M. J. C. Long, R. M. Morrison, P. M. Roberts, E. D. Savory, A. D. Smith, M. J. Sweet and J. M. Withey

Org. Biomol. Chem.2005, DOI 10.1039/b506339f

49. Asymmetric conjugate reductions with samarium diiodide: asymmetric synthesis of (2S,3R)- and (2S,3S)-[2-H,3-2H]-leucine-(S)-phenylalanine dipeptides and (2S,3R)-[2-2H,3-2H]-phenylalanine methyl ester

S. G. Davies, H. Rodriguez-Solla, J. A. Tamayo, A. R. Cowley, C. Concellon, A. Christopher Garner, A. L. Parkes and A. D. Smith

Org. Biomol. Chem.20053, 1435

48. Cyclic β-amino acid derivatives: synthesis via lithium amide promoted tandem asymmetric conjugate addition–cyclisation reactions

S. G. Davies, D. Díez, S. H. Dominguez, N. M. Garrido, D. Kruchinin, P. D. Price and A. D. Smith

Org. Biomol. Chem.20053, 1284

47. A SuperQuat glycolate aldol approach to the asymmetric synthesis of hexose monosaccharides

S. G. Davies, R. L. Nicholson and A D. Smith

Org. Biomol. Chem.20053, 348

46. α-Halo-diketopiperazines as chiral glycine cation equivalents

S. D. Bull, S. G. Davies, A. C. Garner, E. D. Savory, E. J. Snow and A. D. Smith

Tetrahedron: Asymmetry2004, 15, 3989

45. Asymmetric synthesis of 2-alkyl- and 2-aryl-3-aminopropionic acids from (S)-N-acryloyl-5,5-dimethyloxazolidin-2-one derivatives

J. E. Beddow, S. G. Davies, A D. Smith and A. J. Russell

Chem. Commun., 2004, 2778

44. Stereoselective conjugate addition reactions of lithium amides to α,β-unsaturated chiral Iron complexes [(η5-C5H5)Fe(CO)(PPh3)(COCH=CHR)]

J. Dupont, S. G. Davies, R. J. C. Easton, O. Ichihara, J. M. McKenna, A. D. Smith and J. A. A. de Sousa

J. Organomet. Chem., 2004689, 4184

43. Double diastereoselective SuperQuat glycolate aldol reactions; Application to the asymmetric synthesis of polyfunctionalised lactones

S. G. Davies, R. L. Nicholson and A D. Smith

Org. Biomol. Chem.20042, 3385

42. Parallel kinetic resolution oftert-butyl (RS)-3-alkyl cyclopentene-1-carboxylates for the asymmetric synthesis of 3-alkylcispentacin derivatives

S. G. Davies, A. C. Garner, M. J. C. Long, A. D. Smith, M. J. Sweet and J. M. Withey

Org. Biomol. Chem.20042, 3355

41. Kinetic Resolution oftert-butyl (RS)-3-alkylcyclopentene-1-carboxylates for the synthesis of homochiral 3-alkyl cispentacin derivatives

M. E. Bunnage, S. G. Davies, R. M. Parkin, P. M. Roberts, A. D. Smith and J. M. Withey

Org. Biomol. Chem.20042, 3337

40. Highly diastereoselective conjugate reduction with samarium diiodide: synthesis of methyl (2S,3R)-N-acetyl-2-amino-2,3-dideuterio-3-phenylpropionate

S. G. Davies, A. C. Garner, H. Rodríguez-Solla, A. D. Smith and J. A. Tamayo

Chem. Commun., 2004, 2502

39. Asymmetric Synthesis of thecis- andtrans-stereoisomers of 4-aminopyrrolidine-3-carboxylic acid and 4-aminotetrahydrofuran-3-carboxylic acid

M. E. Bunnage, S. G. Davies, P. M. Roberts, A. D. Smith and J. M. Withey

Org. Biomol. Chem.20042, 2763

38. Asymmetric total synthesis of Sperabillins B and Dvialithium amide conjugate addition

S. G. Davies, J. R. Haggitt, O. Ichihara, R. J. Kelly, M. Leech, A. J. Price Mortimer, P. M. Roberts and A. D. Smith

Org. Biomol. Chem.20042, 2630

37. Asymmetric synthesis of 3,4,5,6-tetrasubstituted piperidin-2-ones by three component coupling

S. G. Davies, A. D. Smith and A. R. Cowley

Synlett2004, 1957

36. N-α-benzyloxyoacetyl derivatives of (S)-4-benzyl-5,5-dimethyloxazolidin-2-one for the asymmetric synthesis of differentially protected α,β-dihydroxyaldehydes

S. G. Davies, I. A. Hunter, R. L. Nicholson, P. M. Roberts, E. D. Savory and A. D. Smith

Tetrahedron200460, 7553

35. Asymmetric Synthesis of (4R,5R)-cytoxazone and (4R,5S)-epi-cytoxazone

S. G. Davies, D. G. Hughes, R. L. Nicholson, A. D. Smith and A. J. Wright

Org. Biomol. Chem.2004, 1549

34. Asymmetric synthesis and applications of β-amino Weinreb amides: asymmetric synthesis of (S)-Coniine

A. J. Burke, S. G. Davies, A. C. Garner, T. D. McCarthy, P. M. Roberts, A. D. Smith, H. Rodriguez-Solla and R. J. Vickers

Org. Biomol. Chem.20042, 1387

33. Double asymmetric induction as a mechanistic probe: conjugate addition for the asymmetric synthesis of a pseudotripeptide

S. G. Davies, G. Hermann, A. D. Smith and M. J. Sweet

Chem. Commun., 20041128

32. Iodine mediated ring closing alkene iodoamination with N-debenzylation for the asymmetric synthesis of polyhydroxylated pyrrolidines

S. G. Davies, R. L. Nicholson, P. D. Price, P. M. Roberts and A. D. Smith

Synlett2004, 901

31. Asymmetric synthesis of the stereoisomers of 2-amino-5-carboxymethyl-cyclopentane-1-carboxylate

J. G. Urones, N. M. Garrido, D. Díez, M. M. El Hammouni, S. H. Dominguez, J. A. Casaseca, S. G. Davies and A. D. Smith

Org. Biomol. Chem.20042, 364

30. Preparation of (1R,2S,5S)- and (1S,2R,5R)-methyl 2-amino-5-tert-butyl-cyclopentane-1-carboxylate by parallel kinetic resolution of methyl (±)-5-tert-butyl-cyclopentene-1-carboxylate

S. G. Davies, D. Díez, M. M. El Hammouni, N. M. Garrido, A. C. Garner, M. J. C. Long, R. M. Morrison, A. D. Smith, M. J. Sweet and J. M. Withey

Chem. Commun.2003, 2410.

29. Oxidative functionalisation of SuperQuat enamides: asymmetric synthesis of homochiral 1,2 diols

S. G. Davies, M. Suk-Key, H. R. Solla, H. J. Sanganee, E. D. Savory, A. D. Smith

Synlett, 2003, 1659

28. The Asymmetric Synthesis ofanti-(2S,3S)- andsyn-(2R,3S)-diaminobutanoic acid

M. E. Bunnage, A. J. Burke, S. G. Davies, N. L. Millican, R. L. Nicholson, P. M. Roberts and A. D. Smith

Org. Biomol. Chem.20031, 3708

27. Asymmetric synthesis of (1R,2S,3R)-3-methylcispentacin and (1S,2S,3R)-3-methyltranspentacin by kinetic resolution oftert-butyl (±)-3-methylcyclopentene-1-carboxylate

M. E. Bunnage, A. M. Chippendale, S. G. Davies, R. M. Parkin, A. D. Smith and J. M. Withey

Org. Biomol. Chem.20031, 3698

26. SuperQuatN-acyl-5,5-dimethyl-oxazolidin-2-ones for the asymmetric synthesis of α-alkyl and β-alkyl aldehydes

S. D. Bull, S. G. Davies, R. L. Nicholson, H. J. Sanganee and A. D. Smith

Org. Biomol. Chem.20031, 2886

25. Double diastereoselective aza-Claisen rearrangements

S. G. Davies, A. C. Garner, R. L. Nicholson, J. Osborne, E. D. Savory and A. D. Smith

Chem. Commun., 2003, 2134

24. Asymmetric synthesis of substituted 1-aminocyclopropane-1-carboxylic acidsviadiketopiperazine methodology

E. Bunuel, S. D. Bull, S. G. Davies, A. C. Garner, E. D. Savory, A. D. Smith, R. J. Vickers and D. J. Watkin

Org. Biomol. Chem.20031, 2531

23. N-Acyl-5,5-Dimethyl-oxazolidin-2-ones as Weinreb amide equivalents

J. Bach, S. D. Bull, C. Blachere, S. G. Davies, R. L. Nicholson, P. D. Price, H. J. Sanganee and A. D. Smith

Org. Biomol. Chem., 20031, 2001

22. Asymmetric synthesis of cyclic β-amino acids and cyclic amines via sequential diastereoselective conjugate addition and ring closing metathesis

A. Chippindale, S. G. Davies, K. Iwamoto, R. M. Parkin, C. A. P. Smethurst, A. D. Smith and H. Rodriguez-Solla

Tetrahedron200359, 3253

21. Asymmetric synthesis of (1R,2S,3R)- γ-methyl-cis-pentacin by a kinetic resolution protocol

S. Bailey, S. G. Davies, A. D. Smith and J. M. Withey

Chem. Commun., 2002, 2910 

20. The asymmetric synthesis of D-Galactose via an iterativesyn-glycolate aldol strategy

S. G. Davies, R. L. Nicholson and A. D. Smith

Synlett, 2002, 1637

19. Diastereoselective [2,3] sigmatropic rearrangements ofN-benzyl-O-allylhydroxylamines bearing a stereogenic centre adjacent to the migration terminus

S. D. Bull, S. G. Davies, S. H. Dominguez, S. Jones, T. Sellers, A. J. Price and A. D. Smith

J. Chem. Soc., Perkin Trans. 12002, 2141 

18. Asymmetric synthesis of α-amino carbonyls using lithium (R)-N-benzyl-N-α-methylbenzylamide

S. G. Davies, S. W. Epstein, A. C. Garner, O. Ichihara and A. D. Smith

Tetrahedron: Asymmetry, 200213, 1555

17. Asymmetric synthesis of β-pyridyl-β-amino acid derivatives

S. D. Bull, S. G. Davies, M. Gianotti, P. J. Kelly, E. D. Savory and A. D. Smith

J. Chem. Soc., Perkin Trans. 12002, 1858

16. [2,3] sigmatropic rearrangements of N-benzyl-O-allylhydroxylamines

S. G. Davies, J. F. Fox, S. Jones, M. A. Sanz, A. J. Price, T. Sellers, A. D. Smith and F. C. Teixeira

J. Chem. Soc., Perkin Trans. 12002, 1757 

15. Ring closing metathesis for the asymmetric synthesis of (S)-homopipecolic acid, (S)-homoproline and (S)-coniine

S. G. Davies, K. Iwamoto, C. A. P. Smethurst, A. D. Smith and H. Rodriguez-Solla

Synlett2002, 1146

14. Photochemical incorporation and exchange in mononuclear η5-cyclopentadienyl iron carbonyl complexes

S. G. Davies, S. Jones and A. D. Smith

Trends in Organometallic Chemistry20024, 59

13. Asymmetric synthesis of homochiral differentially protected bis-β-amino acid scaffolds

S. D. Bull, S. G. Davies, P. M. Roberts, E. D. Savory and A. D. Smith

Tetrahedron, 200258, 4629 

12. Asymmetric synthesis of a homochiral differentially protected pseudo-meso bis-β-amino acid scaffold

S. D. Bull, S. G. Davies and A. D. Smith

Tetrahedron: Asymmetry, 200112, 2941

11. Asymmetric synthesis of β-haloaryl β-amino acid derivatives

S. D. Bull, S. G. Davies, S. Delgado-Ballester, M. Gianotti, P. M. Kelly, L. J. Kotchie, M. Laderas and A. D. Smith

J. Chem. Soc., Perkin Trans. 12001, 3112

10. Orthogonal N,N-deprotection strategies of β-amino esters

S. D. Bull, S. G. Davies, M. Gianotti, P. M. Kelly and A. D. Smith

J. Chem. Soc., Perkin Trans. 12001, 3106

9. Asymmetric synthesis of β-amino acid scaffolds

S. D. Bull, S. G. Davies and A. D. Smith

J. Chem. Soc., Perkin Trans. 12001, 2931

8. Asymmetric synthesis of α-amino carbonyls (aldehydes, ketones and acids) using lithium (R)-N-benzyl-N- α-methylbenzylamide

S. G. Davies, S. W. Epstein, O. Ichihara and A. D. Smith

Synlett2001, 1599 

7. Palladium catalysed elaboration Of Codeine and Morphine

S. G. Davies, C. Goodwin, D. Pyatt and A. D. Smith

J. Chem. Soc., Perkin Trans. 12001, 1413

6. Chemoselective oxidative debenzylation ofN-benzyl tertiary amines

S. D. Bull, S. G. Davies, G. Fenton, A. W. Mulvaney, R. S. Prasad and A. D. Smith

J. Chem. Soc., Perkin Trans. 12000, 3765

5. (S)-4-benzyl-5,5-dimethyl-oxazolidin-2-one for the asymmetric synthesis of α-substituted aldehydes

S. D. Bull, S. G. Davies, R. L. Nicholson and A. D. Smith

Tetrahedron: Asymmetry200011, 3475

4. Asymmetric synthesis of β-haloaryl β-amino acid derivatives

S. D. Bull, S. G. Davies, S. Delgado-Ballester, G. Fenton, P. J. Kelly and A. D. Smith

Synlett2000, 1257

3. Asymmetric synthesis of homochiral Baylis-Hillman products employing (R)-N-methyl-N-α-methylbenzyl amide

S. G. Davies, C. A. P. Smethurst, A. D. Smith and G. D. Smyth

Tetrahedron: Asymmetry200011, 2437

2. Chemoselective oxidative debenzylation of tertiaryN-benzyl amines

S. D. Bull, S. G. Davies, G. Fenton, A. W. Mulvaney, R. S. Prasad and A. D. Smith

Chem. Commun., 2000, 337

1. N-Acyl-5,5-dimethyl-oxazolidin-2-ones as latent aldehyde equivalents

J. Bach, S. D. Bull, S. G. Davies, R. L. Nicholson, H. J. Sanganee and A. D. Smith

Tetrahedron Lett.199940, 6677